Challenging targets

Measuring accurate kinetics of compounds on membrane proteins embedded within their native environment (GPCRs, Ion Channels, other receptor classes e.g. ACE)

Intrinsically Discorded Proteins (IDP)

 

Challenging modalities

Fragment screening, covalent fragments, also small molecules, peptides, antibodies, oligonucleotide therapeutics

Detect small or large molecules as biosensing is independent of the molecular weight

We can detect artifacts caused by aggregation and non-specific binding of fragments

 

Protein-Protein Interactions

PPI inhibitors, Induced proximity platforms (PROTAC)

The method is well positioned for screening Protein-Protein Interactions because it works on a 3-body binding problem

Applications